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BRL-15572 dihydrochloride
CAS No. 193611-72-2
BRL-15572 dihydrochloride ( BRL15572;BRL 15572 )
产品货号. M13033 CAS No. 193611-72-2
BRL-15572 is a potent, selective h5-HT1D receptor antagonist.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥332 | 有现货 |
|
| 10MG | ￥535 | 有现货 |
|
| 25MG | ￥875 | 有现货 |
|
| 50MG | ￥1345 | 有现货 |
|
| 100MG | ￥2009 | 有现货 |
|
| 200MG | ￥3021 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称BRL-15572 dihydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述BRL-15572 is a potent, selective h5-HT1D receptor antagonist.
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产品描述BRL-15572 is a potent, selective h5-HT1D receptor antagonist with pKi of 7.9, dispalys 60-fold selectivity over h5-HT1B; shows binding affinities for 5-HT1A, 5-HT1B, 5-HT1E, 5-HT1F, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT6 and 5-HT7 with pKi of 7.7, 6.1, 5.2, 6.0, 6.6, 7.4, 6.2, 5.9 and 6.3, respectively.
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同义词BRL15572;BRL 15572
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT1A; 5-HT1D; 5-HT2A; 5-HT2B; 5-HT7
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研究领域Neurological Disease
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适应症——
化学信息
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CAS Number193611-72-2
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分子量479.87
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分子式C25H29Cl3N2O
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESC1CN(CCN1CC(C(C2=CC=CC=C2)C3=CC=CC=C3)O)C4=CC(=CC=C4)Cl.Cl.Cl
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化学全称1-Piperazineethanol, 4-(3-chlorophenyl)-.alpha.-(diphenylmethyl)-, hydrochloride (1:2)
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Price GW, et al. Naunyn Schmiedebergs Arch Pharmacol. 1997 Sep;356(3):312-20.
2. Schlicker E, et al. Naunyn Schmiedebergs Arch Pharmacol. 1997 Sep;356(3):321-7.
3. De Vries P, et al. Eur J Pharmacol. 1998 Nov 27;362(1):69-72.
4. Marcoli M, et al. Br J Pharmacol. 1999 Feb;126(3):607-12.
2. Schlicker E, et al. Naunyn Schmiedebergs Arch Pharmacol. 1997 Sep;356(3):321-7.
3. De Vries P, et al. Eur J Pharmacol. 1998 Nov 27;362(1):69-72.
4. Marcoli M, et al. Br J Pharmacol. 1999 Feb;126(3):607-12.
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